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TRUTH IN PEPTIDES
Peer Reviewed

Tirzepatide — Interactions & Safety Profile

2 contraindications2 known interactions⚠ Pregnancy warning

Contraindications

Personal or family history of MTC

Same class warning as semaglutide — thyroid C-cell tumour risk in rodents.

MEN 2 syndrome

Predisposition to medullary thyroid carcinoma.

Drug Interactions

Insulin / SulfonylureasSeriousmajor interaction

Increased hypoglycaemia risk.

Reduce insulin or sulfonylurea dose.

Oral contraceptivesModeratemoderate interaction

Delayed gastric emptying may reduce absorption of oral hormonal contraceptives.

Switch to non-oral contraception or use barrier method during dose escalation.

Monitoring Required

  • HbA1c every 3-6 months
  • Signs of pancreatitis
  • Thyroid examination if symptoms develop

Pregnancy & Nursing

Contraindicated. Discontinue ≥2 months before planned pregnancy.

Pending physician review — consult your provider before use.

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